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A convenient preparation of 5-iodo-1,4-disubstituted-1,2,3-triazole: Multicomponent one-pot reaction of azide and alkyne mediated by CuI-NBS
Li, Lingjun1,2; Zhang, Guisheng1; Zhu, Anlian1; Zhang, Lihe2
刊名JOURNAL OF ORGANIC CHEMISTRY
2008-05-02
DOI10.1021/jo800035v
73期:9页:3630-3633
收录类别SCI ; IC ; CCR
文章类型Article
WOS标题词Science & Technology
类目[WOS]Chemistry, Organic
研究领域[WOS]Chemistry
关键词[WOS]CYCLIC ADP-RIBOSE ; CALCIUM-RELEASE ACTIVITY ; CLICK CHEMISTRY ; COPPER(I)-CATALYZED SYNTHESIS ; RAPID SYNTHESIS ; AMINO-ACIDS ; INHIBITORS ; ANALOGS ; 1,2,3-TRIAZOLES ; DISCOVERY
英文摘要

[GRAPHICS]

The system of CuI and NBS was found to provide both I(+) and Cu(+) for the first time. An efficient method for preparation of 5-iodo-1,4-disubstituted-1,2,3-triazole was achieved by multicomponent one-pot reaction of azides with alkynes in the presence of the novel CuI and NBS catalytic system. The high tolerance of various sensitive groups revealed the potential applications of this method in organic synthesis and drug discovery.

语种英语
WOS记录号WOS:000255339600052
引用统计
被引频次:82[WOS]   [WOS记录]     [WOS相关记录]
文献类型期刊论文
条目标识符http://ir.bjmu.edu.cn/handle/400002259/53162
专题北京大学药学院
作者单位1.Henan Normal Univ, Coll Chem & Environm Sci, Xinxiang 453007, Peoples R China
2.Peking Univ, Sch Pharmaceut Sci, Natl Lab Nat & Biomimet Drugs, Beijing 100083, Peoples R China
推荐引用方式
GB/T 7714
Li, Lingjun,Zhang, Guisheng,Zhu, Anlian,et al. A convenient preparation of 5-iodo-1,4-disubstituted-1,2,3-triazole: Multicomponent one-pot reaction of azide and alkyne mediated by CuI-NBS[J]. JOURNAL OF ORGANIC CHEMISTRY,2008,73(9):3630-3633.
APA Li, Lingjun,Zhang, Guisheng,Zhu, Anlian,&Zhang, Lihe.(2008).A convenient preparation of 5-iodo-1,4-disubstituted-1,2,3-triazole: Multicomponent one-pot reaction of azide and alkyne mediated by CuI-NBS.JOURNAL OF ORGANIC CHEMISTRY,73(9),3630-3633.
MLA Li, Lingjun,et al."A convenient preparation of 5-iodo-1,4-disubstituted-1,2,3-triazole: Multicomponent one-pot reaction of azide and alkyne mediated by CuI-NBS".JOURNAL OF ORGANIC CHEMISTRY 73.9(2008):3630-3633.
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