IR@PKUHSC  > 北京大学药学院  > 化学生物学系
学科主题药学
Efficient Preparation of Photolabile Agent MNI-glu by Regioselective Nitration of 4-Methoxyindoline Derivative
Wang, Xiaowei1; Gao, Yu1; Xu, Yang1; Li, Li1; Zhang, Zhili1; Liu, Junyi1,2
关键词Aromatic Nitration Caged L-glutamate Claypop Nitroindolines Photorelease Agent
刊名SYNTHETIC COMMUNICATIONS
2009
DOI10.1080/00397910902883645
39期:22页:4030-4038
收录类别SCI ; CCR
文章类型Article
WOS标题词Science & Technology
类目[WOS]Chemistry, Organic
研究领域[WOS]Chemistry
关键词[WOS]L-GLUTAMATE ; 1-ACYL-7-NITROINDOLINES ; PHOTORELEASE ; PRECURSOR
英文摘要

The present work investigates the nitration of 4-methoxy indoline derivative with different reagents and optimized conditions. We now report a simple methodology for nitration employing claycop in the presence of amine, which offers significant improvement with regard to the yield and regioselectivity, and a much more favorable isomeric ratio of products was obtained under mild conditions. Therefore, a useful method for preparation of a photolabile L-glutamate derivative was concurrently established.

语种英语
WOS记录号WOS:000272207000008
Citation statistics
Cited Times:4[WOS]   [WOS Record]     [Related Records in WOS]
文献类型期刊论文
条目标识符http://ir.bjmu.edu.cn/handle/400002259/55281
Collection北京大学药学院_化学生物学系
作者单位1.Peking Univ, Dept Biol Chem, Sch Pharmaceut Sci, Beijing 100191, Peoples R China
2.Peking Univ, State Key Lab Nat & Biomimet Drugs, Beijing 100191, Peoples R China
Recommended Citation
GB/T 7714
Wang, Xiaowei,Gao, Yu,Xu, Yang,et al. Efficient Preparation of Photolabile Agent MNI-glu by Regioselective Nitration of 4-Methoxyindoline Derivative[J]. SYNTHETIC COMMUNICATIONS,2009,39(22):4030-4038.
APA Wang, Xiaowei,Gao, Yu,Xu, Yang,Li, Li,Zhang, Zhili,&Liu, Junyi.(2009).Efficient Preparation of Photolabile Agent MNI-glu by Regioselective Nitration of 4-Methoxyindoline Derivative.SYNTHETIC COMMUNICATIONS,39(22),4030-4038.
MLA Wang, Xiaowei,et al."Efficient Preparation of Photolabile Agent MNI-glu by Regioselective Nitration of 4-Methoxyindoline Derivative".SYNTHETIC COMMUNICATIONS 39.22(2009):4030-4038.
Files in This Item:
There are no files associated with this item.
Related Services
Recommend this item
Bookmark
Usage statistics
Export to Endnote
谷歌学术
谷歌学术Similar articles in
[Wang, Xiaowei]'s Articles
[Gao, Yu]'s Articles
[Xu, Yang]'s Articles
百度学术
百度学术Similar articles in
[Wang, Xiaowei]'s Articles
[Gao, Yu]'s Articles
[Xu, Yang]'s Articles
必应学术
必应学术Similar articles in
[Wang, Xiaowei]'s Articles
[Gao, Yu]'s Articles
[Xu, Yang]'s Articles
Terms of Use
No data!
Social Bookmark/Share
All comments (0)
No comment.
 

Items in the repository are protected by copyright, with all rights reserved, unless otherwise indicated.