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Efficient Preparation of Photolabile Agent MNI-glu by Regioselective Nitration of 4-Methoxyindoline Derivative
Wang, Xiaowei1; Gao, Yu1; Xu, Yang1; Li, Li1; Zhang, Zhili1; Liu, Junyi1,2
关键词Aromatic Nitration Caged L-glutamate Claypop Nitroindolines Photorelease Agent
刊名SYNTHETIC COMMUNICATIONS
2009
DOI10.1080/00397910902883645
39期:22页:4030-4038
收录类别SCI ; CCR
文章类型Article
WOS标题词Science & Technology
类目[WOS]Chemistry, Organic
资助者National Science Foundation of China ; Ministry of Education of China ; National Science Foundation of China ; Ministry of Education of China
研究领域[WOS]Chemistry
关键词[WOS]L-GLUTAMATE ; 1-ACYL-7-NITROINDOLINES ; PHOTORELEASE ; PRECURSOR
英文摘要

The present work investigates the nitration of 4-methoxy indoline derivative with different reagents and optimized conditions. We now report a simple methodology for nitration employing claycop in the presence of amine, which offers significant improvement with regard to the yield and regioselectivity, and a much more favorable isomeric ratio of products was obtained under mild conditions. Therefore, a useful method for preparation of a photolabile L-glutamate derivative was concurrently established.

语种英语
资助者National Science Foundation of China ; Ministry of Education of China ; National Science Foundation of China ; Ministry of Education of China
WOS记录号WOS:000272207000008
引用统计
被引频次:4[WOS]   [WOS记录]     [WOS相关记录]
文献类型期刊论文
条目标识符http://ir.bjmu.edu.cn/handle/400002259/55281
专题北京大学药学院_化学生物学系
作者单位1.Peking Univ, Dept Biol Chem, Sch Pharmaceut Sci, Beijing 100191, Peoples R China
2.Peking Univ, State Key Lab Nat & Biomimet Drugs, Beijing 100191, Peoples R China
推荐引用方式
GB/T 7714
Wang, Xiaowei,Gao, Yu,Xu, Yang,et al. Efficient Preparation of Photolabile Agent MNI-glu by Regioselective Nitration of 4-Methoxyindoline Derivative[J]. SYNTHETIC COMMUNICATIONS,2009,39(22):4030-4038.
APA Wang, Xiaowei,Gao, Yu,Xu, Yang,Li, Li,Zhang, Zhili,&Liu, Junyi.(2009).Efficient Preparation of Photolabile Agent MNI-glu by Regioselective Nitration of 4-Methoxyindoline Derivative.SYNTHETIC COMMUNICATIONS,39(22),4030-4038.
MLA Wang, Xiaowei,et al."Efficient Preparation of Photolabile Agent MNI-glu by Regioselective Nitration of 4-Methoxyindoline Derivative".SYNTHETIC COMMUNICATIONS 39.22(2009):4030-4038.
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