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学科主题药学
Palladium-Catalyzed Indole and Azaindole Synthesis by Direct Annulation of Electron-Poor o-Chloroanilines and o-Chloroaminopyridines with Aldehydes
Xu, Zhengren; Hu, Weimin; Zhang, Fengying; Li, Qingjiang; Lue, Zhiyao; Zhang, Lihe; Jia, Yanxing
关键词Indole Azaindole Palladium Annulation Ligand
刊名SYNTHESIS-STUTTGART
2008-12-16
DOI10.1055/s-0028-1083225
24页:3981-3987
收录类别SCI ; IC ; CCR
文章类型Article
WOS标题词Science & Technology
类目[WOS]Chemistry, Organic
研究领域[WOS]Chemistry
关键词[WOS]NONREARRANGED MONOTERPENOID UNIT ; HIGHLY FUNCTIONALIZED INDOLES ; SUZUKI-MIYAURA REACTION ; COUPLING REACTIONS ; INTERNAL ALKYNES ; 2,3-DISUBSTITUTED INDOLES ; ALPHA-ARYLATION ; CHLOROPEPTIN-I ; ARYL CHLORIDES ; CYCLIZATION
英文摘要

A practical process for the synthesis of 2-unsubstituted indoles and azaindoles has been developed by the palladium-catalyzed direct annulation of electron-poor o-chloro/bromoanilines and o-chloroaminopyridines with aldehydes. Coupled with the previous results of Jia and Zhu, this allows rapid access to a variety of 2-unsubstituted indoles and azaindoles starting from simple and easily accessible precursors.

语种英语
WOS记录号WOS:000262381500014
Citation statistics
Cited Times:37[WOS]   [WOS Record]     [Related Records in WOS]
文献类型期刊论文
条目标识符http://ir.bjmu.edu.cn/handle/400002259/55452
Collection北京大学药学院
北京大学药学院_药物化学系
作者单位Peking Univ, Sch Pharmaceut Sci, State Key Lab Nat & Biomimet Drugs, Beijing 100191, Peoples R China
Recommended Citation
GB/T 7714
Xu, Zhengren,Hu, Weimin,Zhang, Fengying,et al. Palladium-Catalyzed Indole and Azaindole Synthesis by Direct Annulation of Electron-Poor o-Chloroanilines and o-Chloroaminopyridines with Aldehydes[J]. SYNTHESIS-STUTTGART,2008(24):3981-3987.
APA Xu, Zhengren.,Hu, Weimin.,Zhang, Fengying.,Li, Qingjiang.,Lue, Zhiyao.,...&Jia, Yanxing.(2008).Palladium-Catalyzed Indole and Azaindole Synthesis by Direct Annulation of Electron-Poor o-Chloroanilines and o-Chloroaminopyridines with Aldehydes.SYNTHESIS-STUTTGART(24),3981-3987.
MLA Xu, Zhengren,et al."Palladium-Catalyzed Indole and Azaindole Synthesis by Direct Annulation of Electron-Poor o-Chloroanilines and o-Chloroaminopyridines with Aldehydes".SYNTHESIS-STUTTGART .24(2008):3981-3987.
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