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学科主题: 药学
题名:
Palladium-Catalyzed Indole and Azaindole Synthesis by Direct Annulation of Electron-Poor o-Chloroanilines and o-Chloroaminopyridines with Aldehydes
作者: Xu, Zhengren; Hu, Weimin; Zhang, Fengying; Li, Qingjiang; Lue, Zhiyao; Zhang, Lihe; Jia, Yanxing
关键词: indole ; azaindole ; palladium ; annulation ; ligand
刊名: SYNTHESIS-STUTTGART
发表日期: 2008-12-16
DOI: 10.1055/s-0028-1083225
期: 24, 页:3981-3987
收录类别: SCI ; IC ; CCR
文章类型: Article
WOS标题词: Science & Technology
类目[WOS]: Chemistry, Organic
研究领域[WOS]: Chemistry
关键词[WOS]: NONREARRANGED MONOTERPENOID UNIT ; HIGHLY FUNCTIONALIZED INDOLES ; SUZUKI-MIYAURA REACTION ; COUPLING REACTIONS ; INTERNAL ALKYNES ; 2,3-DISUBSTITUTED INDOLES ; ALPHA-ARYLATION ; CHLOROPEPTIN-I ; ARYL CHLORIDES ; CYCLIZATION
英文摘要:

A practical process for the synthesis of 2-unsubstituted indoles and azaindoles has been developed by the palladium-catalyzed direct annulation of electron-poor o-chloro/bromoanilines and o-chloroaminopyridines with aldehydes. Coupled with the previous results of Jia and Zhu, this allows rapid access to a variety of 2-unsubstituted indoles and azaindoles starting from simple and easily accessible precursors.

语种: 英语
所属项目编号: 20842004
项目资助者: Peking University Health Science Center ; National Natural Science Foundation of China
WOS记录号: WOS:000262381500014
Citation statistics:
内容类型: 期刊论文
URI标识: http://ir.bjmu.edu.cn/handle/400002259/55452
Appears in Collections:北京大学药学院_期刊论文

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作者单位: Peking Univ, Sch Pharmaceut Sci, State Key Lab Nat & Biomimet Drugs, Beijing 100191, Peoples R China

Recommended Citation:
Xu, Zhengren,Hu, Weimin,Zhang, Fengying,et al. Palladium-Catalyzed Indole and Azaindole Synthesis by Direct Annulation of Electron-Poor o-Chloroanilines and o-Chloroaminopyridines with Aldehydes[J]. SYNTHESIS-STUTTGART,2008(24):3981-3987.
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